Galatsis, Paul : rechercher sur Z-Library

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1

Synthesis and SAR comparison of regioisomeric aryl naphthyridines as potent mGlu5 receptor antagonists

Paul Galatsis, Koji Yamagata, John A. Wendt, Cleo J. Connolly, John W. Mickelson, Jared B.J. Milbank, Susan E. Bove, Christopher S. Knauer, Rachel M. Brooker, Corinne E. Augelli-Szafran, Roy D. Schwar

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2007

Langue:

english

Fichier:

PDF, 133 KB

english, 2007

2

Encyclopedia of Reagents for Organic Synthesis || Aluminum Hydride

Année:

2001

Langue:

english

Fichier:

PDF, 96 KB

english, 2001

3

Ligand–Protein Interactions of Selective Casein Kinase 1δ Inhibitors

Mente, Scot, Arnold, Eric, Butler, Todd, Chakrapani, Subramanyam, Chandrasekaran, Ramalakshmi, Cherry, Kevin, DiRico, Ken, Doran, Angela, Fisher, Katherine, Galatsis, Paul, Green, Michael, Hayward, Ma

Journal:

Journal of Medicinal Chemistry

Année:

2013

Langue:

english

Fichier:

PDF, 1.75 MB

english, 2013

4

[Annual Reports in Medicinal Chemistry] Volume 49 || Development of LRRK2 Kinase Inhibitors for Parkinson's Disease

Année:

2014

Langue:

english

Fichier:

PDF, 1.11 MB

english, 2014

5

Leucine-rich repeat kinase 2 inhibitors: a patent review (2014-2016)

Journal:

Expert Opinion on Therapeutic Patents

Année:

2017

Langue:

english

Fichier:

PDF, 1.12 MB

english, 2017

6

Patterning and Templating for Nanoelectronics

Kosmas Galatsis, Kang L. Wang, Mihri Ozkan, Cengiz S. Ozkan, Yu Huang, Jane P. Chang, Harold G. Monbouquette, Yong Chen, Paul Nealey, Youssry Botros

Journal:

Advanced Materials

Année:

2010

Langue:

english

Fichier:

PDF, 1.69 MB

english, 2010

7

ChemInform Abstract: Succinic Acid Amides as P2—P3 Replacements for Inhibitors of Interleukin-1β Converting Enzyme (ICE or Caspase 1).

Paul Galatsis, et al. et al.

Journal:

Année:

2011

Fichier:

PDF, 24 KB

2011

8

ChemInform Abstract: Bradsher Cycloaddition and Bradsher Reaction

Journal:

Année:

2011

Fichier:

PDF, 18 KB

2011

9

ChemInform Abstract: Weiss—Cook Reaction

Journal:

Année:

2011

Fichier:

PDF, 18 KB

2011

10

Construction of fused bicyclic cyclooctane ring frameworks

Paul Galatsis, Jeffrey J Manwell

Journal:

Année:

1995

Langue:

english

Fichier:

PDF, 790 KB

english, 1995

11

Use of iodobenzene diacetate for the synthesis of α-iodoepoxides

Paul Galatsis, Scott D. Millan

Journal:

Tetrahedron Letters

Année:

1991

Langue:

english

Fichier:

PDF, 175 KB

english, 1991

12

Deconjugative aldol-cyclization sequence for the construction of substituted 2-methoxytetrahydrofurans

Paul Galatsis, Jeffrey J. Manwell

Journal:

Tetrahedron Letters

Année:

1995

Langue:

english

Fichier:

PDF, 223 KB

english, 1995

13

Stereochemical consequences in the deprotonation of enoates

Paul Galatsis, Jeffrey J. Manwell, Scott D. Millan

Journal:

Tetrahedron Letters

Année:

1996

Langue:

english

Fichier:

PDF, 182 KB

english, 1996

14

Rational design of 7-arylquinolines as non-competitive metabotropic glutamate receptor subtype 5 antagonists

Jared B.J. Milbank, Christopher S. Knauer, Corinne E. Augelli-Szafran, Annette T. Sakkab-Tan, Kristin K. Lin, Koji Yamagata, Jennifer K. Hoffman, Nian Zhuang, John Thomas, Paul Galatsis, John A. Wendt

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2007

Langue:

english

Fichier:

PDF, 173 KB

english, 2007

15

Carboxylate bioisosteres of pregabalin

Jacob B. Schwarz, Norman L. Colbry, Zhijian Zhu, Brian Nichelson, Nancy S. Barta, Kristin Lin, Raymond A. Hudack, Sian E. Gibbons, Paul Galatsis, Russell J. DeOrazio, David D. Manning, Mark G. Vartani

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2006

Langue:

english

Fichier:

PDF, 120 KB

english, 2006

16

Succinic acid amides as P2–P3 replacements for inhibitors of interleukin-1β converting enzyme (ICE or caspase 1)

Paul Galatsis, Bradley Caprathe, John Gilmore, Anthony Thomas, Kristin Linn, Susan Sheehan, William Harter, Catherine Kostlan, Elizabeth Lunney, Charles Stankovic, John Rubin, Kenneth Brady, Hamish Al

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2010

Langue:

english

Fichier:

PDF, 2.48 MB

english, 2010

17

Inhibition of interleukin-1β converting enzyme (ICE or caspase 1) by aspartyl acyloxyalkyl ketones and aspartyl amidooxyalkyl ketones

Paul Galatsis, Bradley Caprathe, Dennis Downing, John Gilmore, William Harter, Sheryl Hays, Catherine Kostlan, Kristin Linn, Elizabeth Lunney, Kim Para, Anthony Thomas, Joseph Warmus, Hamish Allen, Ke

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2010

Langue:

english

Fichier:

PDF, 2.63 MB

english, 2010

18

Aqueous intermolecular diels-alder chemistry : Reaction of (e)-2,4-pentadienyl ammonium chloride and related ammonium salts with dienophiles in water

Paul A. Grieco, Paul Galatsis, Ronald F. Spohn

Journal:

Année:

1986

Langue:

english

Fichier:

PDF, 660 KB

english, 1986

19

Stereoselective synthesis of substituted oxetanes

Paul Galatsis, Daniel J. Parks

Journal:

Tetrahedron Letters

Année:

1994

Langue:

english

Fichier:

PDF, 248 KB

english, 1994

20

Application of stable isotope labeled glutathione and rapid scanning mass spectrometers in detecting and characterizing reactive metabolites

Abdul Mutlib, Wing Lam, Jim Atherton, Hao Chen, Paul Galatsis, Wayne Stolle

Journal:

Rapid Communications in Mass Spectrometry

Année:

2005

Langue:

english

Fichier:

PDF, 253 KB

english, 2005

21

LC-MS/MS detection of peroxynitrite-derived 3-nitrotyrosine in rat microvessels

John S Althaus, Kari R Schmidt, Scott T Fountain, Michael T Tseng, Richard T Carroll, Paul Galatsis, Edward D Hall

Journal:

Free Radical Biology and Medicine

Année:

2000

Langue:

english

Fichier:

PDF, 442 KB

english, 2000

22

[Tetrahedron Organic Chemistry Series] Palladium in Heterocyclic Chemistry - A Guide for the Synthetic Chemist Volume 26 || Chapter 4 Pyridines

Année:

2007

Langue:

english

Fichier:

PDF, 803 KB

english, 2007

23

Encyclopedia of Reagents for Organic Synthesis || Aluminum Chloride

Année:

2001

Langue:

english

Fichier:

PDF, 93 KB

english, 2001

24

Enantioselective Construction of Cyclic Ethers by An Aldol-Cyclization Sequence

Galatsis, Paul, Millan, Scott D., Ferguson, George

Journal:

Journal of Organic Chemistry

Année:

1997

Langue:

english

Fichier:

PDF, 323 KB

english, 1997

25

Encyclopedia of Reagents for Organic Synthesis || Diisobutylaluminum Hydride

Année:

2001

Langue:

english

Fichier:

PDF, 119 KB

english, 2001

26

Encyclopedia of Reagents for Organic Synthesis || Lithium Tri- tert -butoxyaluminum Hydride

Année:

2001

Langue:

english

Fichier:

PDF, 149 KB

english, 2001

27

1-Alkenylcycloalkoxy radical chemistry. A two-carbon ring expansion methodology

Galatsis, Paul, Millan, Scott D., Faber, Tim

Journal:

Journal of Organic Chemistry

Année:

1993

Langue:

english

Fichier:

PDF, 764 KB

english, 1993

28

4-Hydroxy-2,2,6,6-tetramethylpiperidine-1-oxyl (Tempol) Inhibits Peroxynitrite-Mediated Phenol Nitration

Carroll, Richard T., Galatsis, Paul, Borosky, Susan, Kopec, Karla K., Kumar, Vikram, Althaus, John S., Hall, Edward D.

Journal:

Chemical Research in Toxicology

Année:

2000

Langue:

english

Fichier:

PDF, 146 KB

english, 2000

29

Synthesis of fused-ring cyclobutenones via a tandem [2 + 2] cycloaddition-.beta.-elimination sequence

Galatsis, Paul, Ashbourne, Katherine J., Manwell, Jeffrey J., Wendling, Paula, Dufault, Robert, Hatt, Krista L., Ferguson, George, Gallagher, John F.

Journal:

Journal of Organic Chemistry

Année:

1993

Langue:

english

Fichier:

PDF, 690 KB

english, 1993

30

Functional group manipulation along the perimeter of a hemispherical molecule. Synthesis of dihydro- and tetrahydro-C16-hexaquinacene

Paquette, Leo A., Galatsis, Paul

Journal:

Journal of Organic Chemistry

Année:

1989

Langue:

english

Fichier:

PDF, 587 KB

english, 1989

31

Structures of the germacranolides isoaristolactone and pyroaristolactone

Lange, Gordon L., Galatsis, Paul

Journal:

Journal of Organic Chemistry

Année:

1984

Langue:

english

Fichier:

PDF, 465 KB

english, 1984

32

Tandem Aldol-Cyclization Sequence for the Construction of Cyclic Ethers. The Formation of Substituted Tetrahydrofurans

Galatsis, Paul, Millan, Scott D., Nechala, Patrik, Ferguson, George

Journal:

Journal of Organic Chemistry

Année:

1994

Langue:

english

Fichier:

PDF, 1.27 MB

english, 1994

33

Kinase domain inhibition of leucine rich repeat kinase 2 (LRRK2) using a [1,2,4]triazolo[4,3-b]pyridazine scaffold

Galatsis, Paul, Henderson, Jaclyn L., Kormos, Bethany L., Han, Seungil, Kurumbail, Ravi G., Wager, Travis T., Verhoest, Patrick R., Noell, G. Stephen, Chen, Yi, Needle, Elie, Berger, Zdenek, Steyn, St

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2014

Langue:

english

Fichier:

PDF, 4.56 MB

english, 2014

34

Phosphoproteomic evaluation of pharmacological inhibition of leucine-rich repeat kinase 2 reveals significant off-target effects of LRRK-2-IN-1

Luerman, Gregory C., Nguyen, Chuong, Samaroo, Harry, Loos, Paula, Xi, Hualin, Hurtado-Lorenzo, Andres, Needle, Elie, Stephen Noell, G., Galatsis, Paul, Dunlop, John, Geoghegan, Kieran F., Hirst, Warre

Journal:

Journal of Neurochemistry

Année:

2014

Langue:

english

Fichier:

PDF, 804 KB

english, 2014

35

Discovery of selective 2,4-diaminopyrimidine-based photoaffinity probes for glyoxalase I

Zhou, Yiqing, Guo, Tianlin, Li, Xitao, Dong, Yi, Galatsis, Paul, Johnson, Douglas S., Pan, Zhengying

Journal:

Année:

2014

Langue:

english

Fichier:

PDF, 454 KB

english, 2014

36

Indenone synthesis. Improved synthetic protocol and effect of substitution on the intramolecular Friedel–Crafts acylation

Galatsis, Paul, Manwell, Jeffrey J., Blackwell, James M.

Journal:

Canadian Journal of Chemistry

Année:

1994

Langue:

english

Fichier:

PDF, 323 KB

english, 1994

37

Mass spectrometry of some furanocoumarins

Tang, Sheng-Yuh, Mcgowan, John C., Singh, Marsha, Galatsis, Paul, Ellis, Brian E., Boyd, Robert K., Brown, Stewart A.

Journal:

Canadian Journal of Chemistry

Année:

1979

Langue:

english

Fichier:

PDF, 482 KB

english, 1979

38

[Annual Reports in Medicinal Chemistry] Volume 33 || To Market, To Market - 1997

Année:

1998

Langue:

english

Fichier:

PDF, 3.21 MB

english, 1998

39

[Topics in Medicinal Chemistry] || Leucine-Rich Repeat Kinase 2 (LRRK2) Inhibitors

Année:

2014

Langue:

english

Fichier:

PDF, 1.27 MB

english, 2014

40

Leucine-rich Repeat Kinase 2 (LRRK2) Pharmacological Inhibition Abates α-Synuclein Gene-induced Neurodegeneration

Daher, João P. L., Abdelmotilib, Hisham A., Hu, Xianzhen, Volpicelli-Daley, Laura A., Moehle, Mark S., Fraser, Kyle B., Needle, Elie, Chen, Yi, Steyn, Stefanus J., Galatsis, Paul, Hirst, Warren D., We

Journal:

Journal of Biological Chemistry

Année:

2015

Langue:

english

Fichier:

PDF, 5.08 MB

english, 2015

41

Expedient Construction of the Dicyclopenta[ a , d ]cyclooctene Core of Ceroplastin Di- and Sesterterpenes

Paquette, Leo A., Liang, Shaowo, Galatsis, Paul

Journal:

Année:

1990

Fichier:

PDF, 167 KB

1990

42

Identification and Profiling of a Selective and Brain Penetrant Radioligand for In Vivo Target Occupancy Measurement of Casein Kinase 1 (CK1) Inhibitors

Wager, Travis T, Galatsis, Paul, Chandrasekaran, Ramalakshmi Y., Butler, Todd W, Li, Jianke, Zhang, Lei, Mente, Scot, Subramanyam, Chakrapani, Liu, Shenping, Doran, Angela C, Chang, Cheng, Fisher, Kat

Journal:

ACS Chemical Neuroscience

Année:

2017

Langue:

english

Fichier:

PDF, 2.52 MB

english, 2017

43

[Annual Reports in Medicinal Chemistry] Volume 32 || Chapter 31. To Market, To Market - 1996

Année:

1997

Langue:

english

Fichier:

PDF, 1.35 MB

english, 1997

44

LRRK2 inhibitors induce reversible changes in nonhuman primate lungs without measurable pulmonary deficits

Baptista, Marco A. S., Merchant, Kalpana, Barrett, Ted, Bhargava, Sakshi, Bryce, Dianne K., Ellis, J. Michael, Estrada, Anthony A., Fell, Matthew J., Fiske, Brian K., Fuji, Reina N., Galatsis, Paul, H

Journal:

Science Translational Medicine

Année:

2020

Fichier:

PDF, 3.30 MB

2020